Methyltrienolone increases the aggressiveness and therefore the motivation of the athlet to go to his limits in training. It also decreases the regeneration time. An athlete needs shorter breaks and can train more often. Because methyltrienolone can not be converted into estrogen by the aromatase enzyme due to its structure in the body, unwanted water storage is eliminated. For this reason, methyltrienolone is used for competition preparation or diet.

Methyltrienolone is an orally applicable steroid, which was already developed in the 1960s for use in animal and cell experiments. The synthesis was first described in 1963.Methyltrienolone is one of the strongest oral anabolic steroids ever produced.